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CDK/HDAC-IN-3

CDK/HDAC-IN-3

Item no.	TMO-T78906-25mg
Manufacturer	TargetMol
CASRN	2944087-54-9
Amount	25 mg
Quantity options	100 mg 100 mg 25 mg 25 mg 50 mg 50 mg
Category	Peptides & Proteins Peptides
Type	Peptides
Specific against	other
Smiles	N(C(=O)C1=C(Cl)C=CC=C1Cl)C=2C(C(NC3=CC=C(C(NC4=C(N)C=CC=C4)=O)C=C3)=O)=NNC2
ECLASS 10.1	32160409
ECLASS 11.0	32160409
UNSPSC	12352202
Shipping Condition	Cool pack
Available
Manufacturer - Targets	CDK\|\|\|HDAC
Shipping Temperature	Cool pack
Storage Conditions	-20°C
Molecular Weight	509, 34
Description	CDK/HDAC-IN-3 is an orally active dual inhibitor of HDACs and CDKs, offering potent and selective inhibition of CDK9, CDK12, CDK13, HDAC1, HDAC2, and HDAC3, with IC50 values of 98.32 nM, 98.85 nM, 100 nM, 62.12 nM, 93.28 nM, and 82.87 nM, respectively, and is applicable in the treatment of acute myeloid leukemia (AML) [1].
Pathways	Cell Cycle/Checkpoint\|\|\|Chromatin/Epigenetic\|\|\|DNA Damage/DNA Repair

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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