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AKR1C3-IN-1

AKR1C3-IN-1

Manufacturer	ChemScene
Category	Reagents & Chemicals Molecules
Type	Molecules
Specific against	other
Amount	100mg
Item no.	CS-7878-100mg
eClass 6.1	32169090
eClass 9.0	32169090
Available
CAS	327092-81-9
Purity	>98%
Formula	C16H15NO4S
MWt	317.36
Solubility	DMSO : >= 100 mg/mL (315.10 mM)
Clinical Information	No Development Reported
Pathway	Others
Target	Others
Biological Activity	AKR1C3-IN-1 is a potent, highly selective inhibitor of AKR1C3, with an IC₅₀ of 13 nM. IC50 & Target: IC50: 13 nM (AKR1C3)^[1] In Vitro: AKR1C3-IN-1 shows less potent activities with 20.3+/-3.8 uM against AKR1C1 and >30 uM against AKR1C2 and AKR1C4. AKR1C3-IN-1 inhibits AKR1C3 activity (inhibiting PR-104H formation) with an IC₅₀ of 0.027+/-0.002 uM^[1].

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Amount: 100mg

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Delivery expected until 6/6/2024